YM-254890

Overview
Catalog #	bs-83221c-1mg
Product Name	YM-254890
Specifications
Storage Buffer	White or off-white lyophilize solid
Storage Condition	-20°C
Target
Product Information	YM-254890 is a novel Gαq/11 inhibitor,1 U46619-induced platelet aggregation is inhibited but phorbol ester- or ionophore-induced aggregation is not2 (IC50 = 0.1-0.2 μM)1. It blocks Pasteurella multocida toxin-mediated activation of Gαq.3 A highly useful new tool for studying Gαq/11-coupled receptor signaling and resulting cellular events.4
Description	CAS Number: 568580-02-9 Chemical Name: Gq inhibitor Molecular Weight: 960.10 Formula: C46H69N7O15 Solubility: DMSO (10 mg/ml) Physical Properties: White or off-white lyophilize solid Purity: 95% by HPLC, NMR (Conforms)