GSK6853
| Overview | |
| Catalog # | bs-82758c-5mg |
| Product Name | GSK6853 |
| Specifications | |
| Storage Buffer | White solid |
| Storage Condition | -20°C |
| Target | |
| Product Information | Very potent (pIC50 = 8.6 vs full length protein, 7.7 in cellular assays) inhibitor of Bromodomain and PHD Finger-containing 1 (BRPF1). It displayed >1600-fold selectivity over other bromodomains. |
| Description | CAS Number: 1910124-24-1 Chemical Name: N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide Molecular weight: 409.49 Formula: C22H27N5O3 Solubility: DMSO (25 mg/ml); ethanol (25 mg/ml) Physical Properties: White solid Purity: 98% by HPLC NMR (Conforms) |