Linsitinib
| Overview | |
| Catalog # | bs-83031c-10mg |
| Product Name | Linsitinib |
| Specifications | |
| Storage Buffer | Yellow solid |
| Storage Condition | -20°C |
| Target | |
| Product Information | Linsitinib is a potent and selective dual inhibitor of insulin-like growth factor 1 (IGF-1R) kinase and insulin receptor (InsR) kinase (IC50’s = 35 and 75 nM respectively).1 It has been investigated as a chemotherapeutic in combination with other drugs for various cancers.2-6 |
| Description | CAS Number: 867160-71-2 Chemical Name: 3-[8-Amino-1-(2-phenyl-7-quinolyl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutanol Molecular weight: 421.49 Formula: C26H23N5O Solubility: DMSO (30 mg/ml) Physical Properties: Yellow solid Purity: 98% by HPLC NMR (Conforms) |