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GAC Inhibitor 968

Overview
Catalog # bs-82312c-5mg
Product Name GAC Inhibitor 968
Specifications
Storage Buffer Off-white solid
Storage Condition RT
Target
Product Information Allosteric inhibitor of glutaminase C (GAC).1 Inhibition of GAC blocks oncogenic transformation induced by Rho GTPases in fibroblasts and B lymphoma cells with no effect on normal cells.2 Inhibits liver-type glutaminase GLS2 and suppresses breast tumor growth in vivo.3,4 Reverses acquired erlotinib resistance in non-small cell lung cancer.5
Description CAS Number: 311795-38-7

Chemical Name: 5-(3-bromo-4-(dimethylamino)phenyl)-2,2-dimethyl-2,3,5,6-tetrahydrobenzo[a]-phenanthridin-4(1H)-

Molecular weight: 475.42

Formula: C27H27BrN2O

Solubility: DMSO (11 mg/ml) Ethanol (1 mg/ml)

Physical Properties: Off-white solid

Purity: 98% by TLC NMR (Conforms)

Frequently asked questions

Which applications is GAC Inhibitor 968 (bs-82312C) validated for, and at what dilution?

bs-82312C is validated for Life Science( N/A).

How should bs-82312C be stored?

RT Storage buffer: Off-white solid